Bilastine
Drug Status
Government Approvals
UK(BNF)
WHO Essential Medicine
NO
Known Teratogen
No
Pharmaceutical Class
Antihistamine
Controlled Drug Substance
No
Summary
Bilastine is used to treat allergic rhinitis, which is inflammation of the nasal passages due to allergies, and urticaria, which is a skin rash with itchy welts. It helps reduce symptoms like sneezing, itching, and runny nose.
Bilastine works by blocking histamine receptors, which are parts of cells that react to histamine, a chemical causing allergy symptoms like itching and sneezing. By blocking these receptors, Bilastine prevents these symptoms.
The usual dose of Bilastine for adults is 20 mg once daily. It should be taken orally on an empty stomach, either one hour before or two hours after a meal.
Common side effects of Bilastine include headache and drowsiness, which means feeling sleepy. These effects are generally mild and affect a small percentage of people.
Bilastine may cause drowsiness, so avoid driving until you know how it affects you. It should be used with caution in people with severe kidney problems. Do not take Bilastine if you are allergic to it.
Indications and Purpose
How does Bilastine work?
Bilastine is an antihistamine that works by blocking histamine receptors in the body. Histamine is a chemical released during allergic reactions that causes symptoms like itching, sneezing, and runny nose. By blocking these receptors, Bilastine prevents histamine from causing these symptoms. Think of it like putting a lock on a door to keep unwanted guests out. This action helps relieve allergy symptoms effectively.
Is Bilastine effective?
Bilastine is effective for treating allergic rhinitis, which is inflammation of the nasal passages due to allergies, and urticaria, which is a skin rash with itchy welts. It works by blocking histamine receptors, reducing allergy symptoms like sneezing, itching, and runny nose. Clinical studies show that Bilastine significantly improves these symptoms compared to placebo. It is a reliable option for managing allergy symptoms when taken as directed.
What is Bilastine?
Bilastine is an antihistamine used to treat allergic rhinitis, which is inflammation of the nasal passages due to allergies, and urticaria, which is a skin rash with itchy welts. It works by blocking histamine receptors, reducing symptoms like sneezing, itching, and runny nose. Bilastine is taken orally and provides relief from allergy symptoms without causing significant drowsiness. It's a reliable option for managing allergies.
Directions for Use
For how long do I take Bilastine?
Bilastine is usually taken for short-term relief of allergy symptoms. The duration depends on how long your symptoms last. For seasonal allergies, you might take it during the allergy season. For chronic conditions, your doctor will guide you on how long to continue. Always follow your doctor's advice on the duration of use and consult them if you have any concerns about your treatment plan.
How do I dispose of Bilastine?
Dispose of unused Bilastine by taking it to a drug take-back program or collection site at a pharmacy or hospital. This ensures the medication is disposed of safely and doesn't harm people or the environment. If a take-back program isn't available, you can throw it in the trash at home. Remove it from its original container, mix it with something undesirable like used coffee grounds, seal it in a plastic bag, and throw it away.
How do I take Bilastine?
Take Bilastine once daily on an empty stomach, either one hour before or two hours after a meal. Swallow the tablet whole with water; do not crush it. Avoid grapefruit juice, as it can affect how the medicine works. If you miss a dose, take it as soon as you remember unless it's close to your next dose. In that case, skip the missed dose and continue your regular schedule. Do not take two doses at once. Always follow your doctor's specific instructions for taking Bilastine.
How long does it take for Bilastine to start working?
Bilastine starts working within one to two hours after taking it. You should notice a reduction in allergy symptoms like sneezing and itching fairly quickly. The full therapeutic effect may take a little longer, depending on your body's response and the severity of your symptoms. For best results, take Bilastine as directed by your doctor and continue to monitor your symptoms.
How should I store Bilastine?
Store Bilastine at room temperature, away from moisture and light. Keep it in its original packaging until you're ready to take it. Avoid storing it in humid places like bathrooms, as moisture can affect the medication's effectiveness. Always keep Bilastine out of reach of children to prevent accidental ingestion. Check the expiration date regularly and dispose of any unused or expired medication properly.
What is the usual dose of Bilastine?
The usual dose of Bilastine for adults is 20 mg once daily. This dose is typically taken on an empty stomach, either one hour before or two hours after a meal. There are no specific dose adjustments for children or the elderly, but always follow your doctor's instructions. If you have any concerns about your dose or if adjustments are needed, consult your healthcare provider.
Warnings and Precautions
Can Bilastine be taken safely while breastfeeding?
The safety of Bilastine while breastfeeding is not well-established. It's unclear if Bilastine passes into breast milk or affects milk production. If you're breastfeeding, discuss with your doctor whether Bilastine is the best option for you. They can help weigh the benefits and potential risks, and suggest alternative treatments if necessary to ensure the safety of your baby.
Can Bilastine be taken safely while pregnant?
The safety of Bilastine during pregnancy is not well-established due to limited evidence. Animal studies suggest potential risks, but human data is lacking. If you're pregnant or planning to become pregnant, talk with your doctor about the safest way to manage your allergies. They can help create a treatment plan that considers both your health and your baby's safety.
Can I take Bilastine with other prescription drugs?
Bilastine may interact with other medications that cause drowsiness, such as sedatives or alcohol, increasing the risk of side effects like dizziness. It can also interact with certain antifungal or antibiotic medications, which may affect how Bilastine works. Always inform your doctor about all medications you are taking to avoid potential interactions. They can help adjust your treatment plan to ensure safety and effectiveness.
Does Bilastine have adverse effects?
Adverse effects are unwanted reactions to a medication. With Bilastine, common adverse effects include headache and drowsiness, affecting a small percentage of users. Serious adverse effects are rare but can include allergic reactions like rash or swelling. If you experience any new or worsening symptoms, contact your doctor. They can help determine if these symptoms are related to Bilastine and advise on the best course of action.
Does Bilastine have any safety warnings?
Bilastine has some safety warnings you should be aware of. It may cause drowsiness, so avoid driving or operating heavy machinery until you know how it affects you. Bilastine should be used with caution in people with severe kidney problems. Not adhering to these warnings can lead to increased side effects or reduced effectiveness of the medication. Always follow your doctor's advice and report any unusual symptoms.
Is Bilastine addictive?
Bilastine is not addictive or habit-forming. It does not cause dependency or withdrawal symptoms when you stop taking it. Bilastine works by blocking histamine receptors to relieve allergy symptoms, and this mechanism does not affect brain chemistry in ways that could lead to addiction. You won't experience cravings for this medication or feel compelled to take more than prescribed. If you have concerns about medication dependence, you can feel confident that Bilastine doesn't carry this risk.
Is Bilastine safe for the elderly?
Elderly individuals may be more sensitive to the effects of Bilastine, particularly drowsiness. This can increase the risk of falls or accidents. Bilastine is generally safe for the elderly, but it's important to start with the lowest effective dose and monitor for side effects. Regular check-ins with a healthcare provider can help ensure the medication is working safely and effectively.
Is it safe to drink alcohol while taking Bilastine?
It's best to avoid alcohol while taking Bilastine. Alcohol can increase the sedative effects of Bilastine, leading to increased drowsiness or dizziness. This can impair your ability to perform tasks that require alertness, like driving. If you choose to drink, do so in moderation and be aware of how your body responds. Talk with your doctor about alcohol use while taking Bilastine for personalized advice.
Is it safe to exercise while taking Bilastine?
You can exercise while taking Bilastine, but be mindful of its potential to cause drowsiness. This might affect your coordination or energy levels during physical activity. To exercise safely, start with light activities and see how your body responds. If you feel dizzy or unusually tired, take a break and rest. Most people can maintain their regular exercise routine while taking Bilastine, but consult your doctor if you have concerns.
Is it safe to stop Bilastine?
Bilastine is often used for temporary relief of allergy symptoms, so you can stop taking it once your symptoms improve. There are no withdrawal symptoms associated with stopping Bilastine. However, if you stop taking it too soon, your allergy symptoms may return. Always follow your doctor's advice on how long to take Bilastine and consult them if you have any concerns about stopping the medication.
What are the most common side effects of Bilastine?
Side effects are unwanted reactions that can occur with medication use. For Bilastine, common side effects include headache and drowsiness. These effects are generally mild and affect a small percentage of people. If you experience new symptoms after starting Bilastine, they might be temporary or unrelated to the medication. Always talk with your doctor before stopping any medication to ensure it's safe to do so.
Who should avoid taking Bilastine?
Do not take Bilastine if you are allergic to it or any of its ingredients. Serious allergic reactions, which cause rash, hives, or swelling that makes breathing difficult, require immediate medical help. Use caution if you have severe kidney problems, as Bilastine may not be suitable for you. Always consult your doctor about any health conditions or medications you are taking to ensure Bilastine is safe for you.